Drugs target to DPYD

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
GIMERACILSmall moleculehead and neck malignant neoplasiaDihydropyrimidine dehydrogenase inhibitor3.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor2.0Active, not recruitingClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculepancreatic ductal adenocarcinomaDihydropyrimidine dehydrogenase inhibitor1.0RecruitingClinicalTrials
GIMERACILSmall moleculebreast neoplasmDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculebiliary tract cancerDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculestomach neoplasmDihydropyrimidine dehydrogenase inhibitor3.0RecruitingClinicalTrials
GIMERACILSmall moleculecolorectal carcinomaDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculenasopharyngeal neoplasmDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculemetastatic colorectal cancerDihydropyrimidine dehydrogenase inhibitor3.0SuspendedClinicalTrials
GIMERACILSmall moleculepancreatic adenocarcinomaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculegastric carcinomaDihydropyrimidine dehydrogenase inhibitor1.0Unknown statusClinicalTrials
GIMERACILSmall moleculecolorectal cancerDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
GIMERACILSmall moleculecolorectal neoplasmDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastroesophageal junction adenocarcinomaDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculeesophageal cancerDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor1.0Active, not recruitingClinicalTrials
GIMERACILSmall moleculestomach neoplasmDihydropyrimidine dehydrogenase inhibitor2.0Active, not recruitingClinicalTrials
GIMERACILSmall moleculeDigestive System CarcinomaDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculeesophageal carcinomaDihydropyrimidine dehydrogenase inhibitor3.0Unknown statusClinicalTrials
GIMERACILSmall moleculenon-small cell lung carcinomaDihydropyrimidine dehydrogenase inhibitor1.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor2.0SuspendedClinicalTrials
GIMERACILSmall moleculecancerDihydropyrimidine dehydrogenase inhibitor2.0TerminatedClinicalTrials
GIMERACILSmall moleculenasopharyngeal neoplasmDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculeneoplasmDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculestomach neoplasmDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor1.0RecruitingClinicalTrials
GIMERACILSmall moleculecervical cancerDihydropyrimidine dehydrogenase inhibitor1.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculestomach neoplasmDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculecolorectal adenocarcinomaDihydropyrimidine dehydrogenase inhibitor3.0RecruitingClinicalTrials
GIMERACILSmall moleculehepatocellular carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor1.0SuspendedClinicalTrials
GIMERACILSmall moleculebreast cancerDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor2.0TerminatedClinicalTrials
GIMERACILSmall moleculenon-small cell lung carcinomaDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculebiliary tract cancerDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculeesophageal squamous cell carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor3.0TerminatedClinicalTrials
ENILURACILSmall moleculecancerDihydropyrimidine dehydrogenase inhibitor1.0RecruitingClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor1.0TerminatedClinicalTrials
GIMERACILSmall moleculebiliary tract cancerDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculehead and neck malignant neoplasiaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculecolorectal neoplasmDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculecolorectal neoplasmDihydropyrimidine dehydrogenase inhibitor2.0WithdrawnClinicalTrials
GIMERACILSmall moleculerectal carcinomaDihydropyrimidine dehydrogenase inhibitor1.0Unknown statusClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor4.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculestomach neoplasmDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
ENILURACILSmall moleculecolorectal adenocarcinomaDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
GIMERACILSmall moleculesecondary malignant neoplasmDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor3.0Unknown statusClinicalTrials
GIMERACILSmall moleculebreast neoplasmDihydropyrimidine dehydrogenase inhibitor4.0Unknown statusClinicalTrials
ENILURACILSmall moleculerectum cancerDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
GIMERACILSmall moleculeesophageal squamous cell carcinomaDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculeesophageal adenocarcinomaDihydropyrimidine dehydrogenase inhibitor1.0RecruitingClinicalTrials
GIMERACILSmall moleculenasopharyngeal neoplasmDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculecolorectal adenocarcinomaDihydropyrimidine dehydrogenase inhibitor3.0WithdrawnClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor2.0TerminatedClinicalTrials
GIMERACILSmall moleculegastroesophageal junction adenocarcinomaDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculerectum cancerDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculecolorectal carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculehepatocellular carcinomaDihydropyrimidine dehydrogenase inhibitor2.0WithdrawnClinicalTrials
GIMERACILSmall moleculerectum cancerDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculenon-small cell lung carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculeneuroendocrine carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor1.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculepancreatic neoplasmDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor1.0Unknown statusClinicalTrials
GIMERACILSmall moleculemetastatic colorectal cancerDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculehepatocellular carcinomaDihydropyrimidine dehydrogenase inhibitor4.0Unknown statusClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculecolorectal carcinomaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculebiliary tract cancerDihydropyrimidine dehydrogenase inhibitor2.0Active, not recruitingClinicalTrials
GIMERACILSmall moleculehead and neck malignant neoplasiaDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculeesophageal cancerDihydropyrimidine dehydrogenase inhibitor3.0RecruitingClinicalTrials
GIMERACILSmall moleculeadenocarcinomaDihydropyrimidine dehydrogenase inhibitor3.0RecruitingClinicalTrials
ENILURACILSmall moleculemalignant colon neoplasmDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
GIMERACILSmall moleculeneoplasmDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
ENILURACILSmall moleculehead and neck malignant neoplasiaDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculegastric adenocarcinomaDihydropyrimidine dehydrogenase inhibitor1.0TerminatedClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculemetastatic colorectal cancerDihydropyrimidine dehydrogenase inhibitor1.0WithdrawnClinicalTrials
ENILURACILSmall moleculelymphomaDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor3.0RecruitingClinicalTrials
GIMERACILSmall moleculehead and neck squamous cell carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
ENILURACILSmall moleculecolorectal carcinomaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculenon-small cell lung carcinomaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculeesophageal squamous cell carcinomaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculestomach neoplasmDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
ENILURACILSmall moleculecolorectal carcinomaDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculecholangiocarcinomaDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
GIMERACILSmall moleculebiliary tract cancerDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculepancreatic ductal adenocarcinomaDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor2.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculesmall cell lung carcinomaDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculecolorectal carcinomaDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
GIMERACILSmall moleculeesophageal cancerDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
ENILURACILSmall moleculebreast cancerDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor3.0WithdrawnClinicalTrials
GIMERACILSmall moleculeesophageal cancerDihydropyrimidine dehydrogenase inhibitor1.0CompletedClinicalTrials
GIMERACILSmall moleculeesophageal cancerDihydropyrimidine dehydrogenase inhibitor2.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor3.0Active, not recruitingClinicalTrials
GIMERACILSmall moleculehead and neck squamous cell carcinomaDihydropyrimidine dehydrogenase inhibitor2.0CompletedClinicalTrials
GIMERACILSmall moleculegastric adenocarcinomaDihydropyrimidine dehydrogenase inhibitor2.0RecruitingClinicalTrials
GIMERACILSmall moleculepancreatic carcinomaDihydropyrimidine dehydrogenase inhibitor1.0SuspendedClinicalTrials
GIMERACILSmall moleculeesophageal squamous cell carcinomaDihydropyrimidine dehydrogenase inhibitor2.0Active, not recruitingClinicalTrials
GIMERACILSmall moleculegastric adenocarcinomaDihydropyrimidine dehydrogenase inhibitor3.0Unknown statusClinicalTrials
GIMERACILSmall moleculegastric carcinomaDihydropyrimidine dehydrogenase inhibitor3.0Not yet recruitingClinicalTrials
GIMERACILSmall moleculegastric cancerDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials
GIMERACILSmall moleculestomach neoplasmDihydropyrimidine dehydrogenase inhibitor3.0CompletedClinicalTrials