Drugs target to AURKB

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
IBCASERTIBSmall moleculetriple-negative breast cancerSerine/threonine-protein kinase Aurora-B inhibitor2.0RecruitingClinicalTrials
IBCASERTIBSmall moleculenon-Hodgkins lymphomaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
IBCASERTIBSmall moleculesmall cell lung carcinomaSerine/threonine-protein kinase Aurora-B inhibitor3.0RecruitingClinicalTrials
ENMD-2076Small moleculehepatocellular carcinomaSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
ENMD-2076Small moleculelymphoid neoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TOZASERTIBSmall moleculemyelodysplastic syndromeSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
MK-6592Small moleculeneoplasmSerine/threonine-protein kinase Aurora inhibitor1.0TerminatedClinicalTrials
SNS-314Small moleculeneoplasmSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
BARASERTIBSmall moleculelymphomaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
BARASERTIBSmall moleculeneoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0TerminatedClinicalTrials
TAK-901Small moleculeacute myeloid leukemiaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TTP-607Small moleculecancerSerine/threonine-protein kinase Aurora inhibitor1.0WithdrawnClinicalTrials
ENMD-2076Small moleculebreast cancerSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
IBCASERTIBSmall moleculeovarian cancerSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
KW-2449Small moleculeacute myeloid leukemiaSerine/threonine-protein kinase Aurora-B inhibitor1.0TerminatedClinicalTrials
IBCASERTIBSmall moleculeovarian cancerSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
BARASERTIBSmall moleculeacute myeloid leukemiaSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
TTP-607Small moleculelymphomaSerine/threonine-protein kinase Aurora inhibitor1.0WithdrawnClinicalTrials
CYC-116Small moleculeneoplasmSerine/threonine-protein kinase Aurora inhibitor1.0TerminatedClinicalTrials
IBCASERTIBSmall moleculesmall cell lung carcinomaSerine/threonine-protein kinase Aurora-B inhibitor1.0RecruitingClinicalTrials
ENMD-2076Small moleculeovarian cancerSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
TOZASERTIBSmall moleculechronic myelogenous leukemiaSerine/threonine-protein kinase Aurora inhibitor1.0TerminatedClinicalTrials
AT-9283Small moleculeneoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TOZASERTIBSmall moleculenon-small cell lung carcinomaSerine/threonine-protein kinase Aurora inhibitor2.0TerminatedClinicalTrials
BI-811283Small moleculeneoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
DANUSERTIBSmall moleculeleukemiaSerine/threonine-protein kinase Aurora inhibitor2.0Unknown statusClinicalTrials
IBCASERTIBSmall moleculeovarian cancerSerine/threonine-protein kinase Aurora-B inhibitor3.0RecruitingClinicalTrials
TOZASERTIBSmall moleculecancerSerine/threonine-protein kinase Aurora inhibitor1.0TerminatedClinicalTrials
ILORASERTIBSmall moleculemetastatic malignant neoplasmSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
ENMD-2076Small moleculemultiple myelomaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
DANUSERTIBSmall moleculeprostate cancerSerine/threonine-protein kinase Aurora inhibitor2.0CompletedClinicalTrials
BARASERTIBSmall moleculeneoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
ILORASERTIBSmall moleculecancerSerine/threonine-protein kinase Aurora inhibitor2.0CompletedClinicalTrials
TOZASERTIBSmall moleculecolorectal carcinomaSerine/threonine-protein kinase Aurora inhibitor1.0TerminatedClinicalTrials
ENMD-2076Small moleculeclear cell adenocarcinomaSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
TAK-901Small moleculemyelodysplastic syndromeSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
BARASERTIBSmall moleculeacute myeloid leukemiaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TOZASERTIBSmall moleculechronic myelogenous leukemiaSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
AT-9283Small moleculenon-Hodgkins lymphomaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TOZASERTIBSmall moleculeacute lymphoblastic leukemiaSerine/threonine-protein kinase Aurora inhibitor1.0TerminatedClinicalTrials
BARASERTIBSmall moleculemyeloid leukemiaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
ENMD-2076Small moleculeFallopian Tube CarcinomaSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
ENMD-2076Small moleculecancerSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
DANUSERTIBSmall moleculemultiple myelomaSerine/threonine-protein kinase Aurora inhibitor2.0TerminatedClinicalTrials
IBCASERTIBSmall moleculeneoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TOZASERTIBSmall moleculelymphoid leukemiaSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
ENMD-2076Small moleculeperitoneum cancerSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
CENISERTIBSmall moleculelymphoid neoplasmSerine/threonine-protein kinase Aurora inhibitor1.0TerminatedClinicalTrials
TAK-901Small moleculemyelofibrosisSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
IBCASERTIBSmall moleculesoft tissue sarcomaSerine/threonine-protein kinase Aurora-B inhibitor2.0RecruitingClinicalTrials
AMG-900Small moleculemyeloid leukemiaSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
TAK-901Small moleculechronic lymphocytic leukemiaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
AMG-900Small moleculecancerSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
CENISERTIBSmall moleculeneoplasmSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
ENMD-2076Small moleculesoft tissue sarcomaSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
TAK-901Small moleculeprimary myelofibrosisSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
PF-03814735Small moleculeneoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
BI-811283Small moleculeacute myeloid leukemiaSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
TOZASERTIBSmall moleculeleukemiaSerine/threonine-protein kinase Aurora inhibitor2.0TerminatedClinicalTrials
AT-9283Small moleculemultiple myelomaSerine/threonine-protein kinase Aurora-B inhibitor2.0CompletedClinicalTrials
GSK-1070916Small moleculeneoplasmSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
IBCASERTIBSmall moleculenon-Hodgkins lymphomaSerine/threonine-protein kinase Aurora-B inhibitor1.0TerminatedClinicalTrials
IBCASERTIBSmall moleculehepatocellular carcinomaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TAK-901Small moleculelymphomaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TAK-901Small moleculemultiple myelomaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
TAK-901Small moleculeWaldenstrom macroglobulinemiaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials
ILORASERTIBSmall moleculeneoplasmSerine/threonine-protein kinase Aurora inhibitor1.0CompletedClinicalTrials
AT-9283Small moleculeleukemiaSerine/threonine-protein kinase Aurora-B inhibitor1.0CompletedClinicalTrials