Drugs target to ATR

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
CERALASERTIBSmall moleculebreast carcinomaSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculemetastatic colorectal cancerSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculeprostate cancerSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculebreast neoplasmSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculeFallopian Tube CarcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculeoral squamous cell carcinomaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculemetastatic prostate cancerSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculenon-small cell lung carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculenon-small cell lung carcinomaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
ELIMUSERTIBSmall moleculeovarian cancerSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculehead and neck squamous cell carcinomaSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials
CERALASERTIBSmall moleculecarcinomaSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculesmall cell lung carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculesmall cell lung carcinomaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
ELIMUSERTIBSmall moleculeMantle cell lymphomaSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculecancerSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculemelanomaSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
CERALASERTIBSmall moleculebreast cancerSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculeureter urothelial carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
M4344Small moleculeovarian cancerSerine-protein kinase ATR inhibitor1.0Not yet recruitingClinicalTrials
CERALASERTIBSmall moleculeneoplasmSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
M4344Small moleculeneoplasmSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials
CERALASERTIBSmall moleculebile duct cancerSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculeneoplasmSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculesmall cell lung carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculesquamous cell carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculebreast cancerSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
M4344Small moleculebreast cancerSerine-protein kinase ATR inhibitor1.0WithdrawnClinicalTrials
BERZOSERTIBSmall moleculebladder transitional cell carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculebreast cancerSerine-protein kinase ATR inhibitor2.0Not yet recruitingClinicalTrials
CERALASERTIBSmall moleculeosteosarcomaSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculeovarian neoplasmSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculehypopharyngeal squamous cell carcinomaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculeneoplasmSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculecancerSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculemetastatic malignant neoplasmSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculenon-small cell lung carcinomaSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculecolorectal adenocarcinomaSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculesmall cell lung carcinomaSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculepancreatic carcinomaSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculecancerSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculeneoplasmSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials
ELIMUSERTIBSmall moleculemetastatic malignant neoplasmSerine-protein kinase ATR inhibitor1.0WithdrawnClinicalTrials
CERALASERTIBSmall moleculeovarian cancerSerine-protein kinase ATR inhibitor2.0WithdrawnClinicalTrials
BERZOSERTIBSmall moleculelaryngeal squamous cell carcinomaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculeoropharynx squamous cell carcinomaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculeprimary peritoneal carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculeadenocarcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculechronic lymphocytic leukemiaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
BERZOSERTIBSmall moleculebreast carcinomaSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculeprolymphocytic leukemiaSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials
BERZOSERTIBSmall moleculesmall cell lung carcinomaSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculeovarian carcinomaSerine-protein kinase ATR inhibitor2.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculeneoplasmSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculecancerSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials
BERZOSERTIBSmall moleculeovarian cancerSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials
CERALASERTIBSmall moleculesmall cell lung carcinomaSerine-protein kinase ATR inhibitor2.0CompletedClinicalTrials
BERZOSERTIBSmall moleculeleiomyosarcomaSerine-protein kinase ATR inhibitor2.0RecruitingClinicalTrials
BERZOSERTIBSmall moleculecervical adenocarcinomaSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculeneoplasmSerine-protein kinase ATR inhibitor1.0Unknown statusClinicalTrials
CERALASERTIBSmall moleculechronic lymphocytic leukemiaSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials
BERZOSERTIBSmall moleculenon-small cell lung carcinomaSerine-protein kinase ATR inhibitor1.0RecruitingClinicalTrials
CERALASERTIBSmall moleculenon-small cell lung carcinomaSerine-protein kinase ATR inhibitor3.0RecruitingClinicalTrials
ELIMUSERTIBSmall moleculeneoplasmSerine-protein kinase ATR inhibitor1.0Active, not recruitingClinicalTrials
CERALASERTIBSmall moleculediffuse large B-cell lymphomaSerine-protein kinase ATR inhibitor1.0CompletedClinicalTrials