Drugs target to TNKS

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
2X-121Small moleculeneoplasmTankyrase 1/2 inhibitor1.0RecruitingClinicalTrials
2X-121Small moleculebreast carcinomaTankyrase 1/2 inhibitor1.0WithdrawnClinicalTrials
2X-121Small moleculebreast cancerTankyrase 1/2 inhibitor2.0Active, not recruitingClinicalTrials
2X-121Small moleculeovarian cancerTankyrase 1/2 inhibitor2.0RecruitingClinicalTrials