Drugs target to TUBA1A

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
PACLITAXEL POLIGLUMEXSmall moleculenon-small cell lung carcinomaTubulin stabiliser2.0CompletedClinicalTrials
T-900607Small moleculeovarian neoplasmTubulin disrupting agent2.0Unknown statusClinicalTrials
DAVUNETIDEProteinCognitive impairmentTubulin stabiliser2.0CompletedClinicalTrials
FOSBRETABULINSmall moleculeovarian cancerTubulin inhibitor2.0TerminatedClinicalTrials
DOLASTATIN-10Small moleculekidney cancerTubulin inhibitor2.0CompletedClinicalTrials
DOLASTATIN-10Small moleculesarcomaTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculenon-small cell lung carcinomaTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculeurogenital neoplasmTubulin inhibitor3.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculesquamous cell carcinomaTubulin stabiliser1.0CompletedClinicalTrials
SOBLIDOTINSmall moleculesarcomaTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculehead and neck carcinomaTubulin inhibitor3.0CompletedClinicalTrials
SAGOPILONESmall moleculeneoplasmTubulin stabiliser1.0CompletedClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodyneoplasmTubulin inhibitor1.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculePrimary Peritoneal Serous AdenocarcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeovarian cancerTubulin stabiliser1.0CompletedClinicalTrials
TUSAMITAMAB RAVTANSINEAntibodyneoplasmTubulin inhibitor1.0Active, not recruitingClinicalTrials
SOBLIDOTINSmall moleculelung cancerTubulin inhibitor2.0CompletedClinicalTrials
ANG1005Proteinglioblastoma multiformeTubulin inhibitor2.0CompletedClinicalTrials
DOLASTATIN-10Small moleculemalignant tumor of extrahepatic bile ductTubulin inhibitor2.0CompletedClinicalTrials
TUSAMITAMAB RAVTANSINEAntibodynon-small cell lung carcinomaTubulin inhibitor3.0RecruitingClinicalTrials
DAVUNETIDEProteinprogressive supranuclear palsyTubulin stabiliser2.0CompletedClinicalTrials
T-900607Small moleculehepatocellular carcinomaTubulin disrupting agent2.0Unknown statusClinicalTrials
T-900607Small moleculenon-Hodgkins lymphomaTubulin disrupting agent2.0TerminatedClinicalTrials
FOSBRETABULINSmall moleculewet macular degenerationTubulin inhibitor1.0CompletedClinicalTrials
FOSBRETABULIN DISODIUMSmall moleculehead and neck malignant neoplasiaTubulin inhibitor2.0CompletedClinicalTrials
FOSBRETABULINSmall moleculehead and neck malignant neoplasiaTubulin inhibitor1.0TerminatedClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodyEndometrial Clear Cell AdenocarcinomaTubulin inhibitor2.0WithdrawnClinicalTrials
VINFLUNINESmall moleculesmall cell lung carcinomaTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculeurogenital neoplasmTubulin inhibitor3.0RecruitingClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculenon-small cell lung carcinomaTubulin stabiliser3.0TerminatedClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodyprimary peritoneal carcinomaTubulin inhibitor1.0CompletedClinicalTrials
MILATAXELSmall moleculecolonic neoplasmTubulin inhibitor2.0CompletedClinicalTrials
ARX-788Unknownbreast cancerTubulin inhibitor2.0RecruitingClinicalTrials
ARX-788Unknowntriple-negative breast cancerTubulin inhibitor2.0RecruitingClinicalTrials
VINFLUNINESmall moleculeurinary bladder cancerTubulin inhibitor3.0CompletedClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodyovarian cancerTubulin inhibitor1.0CompletedClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodymultiple myelomaTubulin inhibitor1.0CompletedClinicalTrials
FOSBRETABULINSmall moleculecancerTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculelung cancerTubulin inhibitor2.0TerminatedClinicalTrials
VINFLUNINESmall moleculeurothelial carcinomaTubulin inhibitor3.0CompletedClinicalTrials
FOSBRETABULIN DISODIUMSmall moleculecancerTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculeprostate cancerTubulin inhibitor2.0CompletedClinicalTrials
DOLASTATIN-10Small moleculeleukemiaTubulin inhibitor2.0CompletedClinicalTrials
PLINABULINSmall moleculenon-small cell lung carcinomaTubulin inhibitor1.0Active, not recruitingClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeprostate adenocarcinomaTubulin stabiliser2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeMalignant Ovarian Brenner TumorTubulin stabiliser3.0Active, not recruitingClinicalTrials
TUSAMITAMAB RAVTANSINEAntibodynon-small cell lung carcinomaTubulin inhibitor2.0RecruitingClinicalTrials
FOSBRETABULINSmall moleculeneuroendocrine neoplasmTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculecancerTubulin inhibitor1.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeovarian clear cell adenocarcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculebreast cancerTubulin stabiliser2.0WithdrawnClinicalTrials
SAGOPILONESmall moleculeglioblastoma multiformeTubulin stabiliser2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeovarian serous adenocarcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeperitoneum cancerTubulin stabiliser1.0CompletedClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodysmall cell lung carcinomaTubulin inhibitor1.0TerminatedClinicalTrials
SAGOPILONESmall moleculenon-small cell lung carcinomaTubulin stabiliser2.0CompletedClinicalTrials
SAGOPILONESmall moleculeprostate cancerTubulin stabiliser2.0CompletedClinicalTrials
TUSAMITAMAB RAVTANSINEAntibodyneoplasmTubulin inhibitor1.0RecruitingClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculenon-small cell lung carcinomaTubulin stabiliser2.0TerminatedClinicalTrials
FOSBRETABULIN DISODIUMSmall moleculewet macular degenerationTubulin inhibitor1.0CompletedClinicalTrials
PLINABULINSmall moleculenon-small cell lung carcinomaTubulin inhibitor3.0CompletedClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodyEndometrial Serous AdenocarcinomaTubulin inhibitor2.0WithdrawnClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodyneuroblastomaTubulin inhibitor2.0CompletedClinicalTrials
PLOCABULINSmall moleculecolorectal cancerTubulin inhibitor2.0CompletedClinicalTrials
PLOCABULINSmall moleculeneoplasmTubulin inhibitor1.0CompletedClinicalTrials
FOSBRETABULINSmall moleculethyroid cancerTubulin inhibitor3.0WithdrawnClinicalTrials
VINFLUNINESmall moleculepenile neoplasmTubulin inhibitor2.0CompletedClinicalTrials
SAGOPILONESmall moleculebreast neoplasmTubulin stabiliser2.0CompletedClinicalTrials
ARX-788Unknownbreast neoplasmTubulin inhibitor1.0TerminatedClinicalTrials
PLINABULINSmall moleculemultiple myelomaTubulin inhibitor2.0RecruitingClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeFallopian Tube Serous AdenocarcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
FOSBRETABULINSmall moleculeneuroendocrine neoplasmTubulin inhibitor1.0TerminatedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculebreast cancerTubulin stabiliser2.0CompletedClinicalTrials
CROLIBULINSmall moleculethyroid cancerTubulin inhibitor1.0CompletedClinicalTrials
INDIBULINSmall moleculecancerTubulin inhibitor1.0CompletedClinicalTrials
DOLASTATIN-10Small moleculeovarian cancerTubulin inhibitor2.0CompletedClinicalTrials
OMBRABULINSmall moleculeovarian cancerTubulin inhibitor2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculefallopian tube cancerTubulin stabiliser1.0CompletedClinicalTrials
SAGOPILONESmall moleculesmall cell lung carcinomaTubulin stabiliser2.0TerminatedClinicalTrials
DAVUNETIDEProteinschizophreniaTubulin stabiliser2.0CompletedClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodyPleuropulmonary blastomaTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculeneoplasmTubulin inhibitor4.0-ATC
FOSBRETABULIN DISODIUMSmall moleculehead and neck malignant neoplasiaTubulin inhibitor1.0TerminatedClinicalTrials
T-900607Small moleculegastric cancerTubulin disrupting agent2.0CompletedClinicalTrials
FOSBRETABULINSmall moleculeovarian cancerTubulin inhibitor1.0TerminatedClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodyleukemiaTubulin inhibitor2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeundifferentiated carcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
VINFLUNINESmall moleculebreast cancerTubulin inhibitor3.0CompletedClinicalTrials
PRALUZATAMAB RAVTANSINEAntibodybreast cancerTubulin inhibitor2.0Active, not recruitingClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodyfallopian tube cancerTubulin inhibitor1.0CompletedClinicalTrials
VERUBULINSmall moleculeneoplasmTubulin disrupting agent1.0CompletedClinicalTrials
MILATAXELSmall moleculerectum cancerTubulin inhibitor2.0CompletedClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodyrhabdomyosarcomaTubulin inhibitor2.0CompletedClinicalTrials
ANG1005Proteinmalignant gliomaTubulin inhibitor1.0CompletedClinicalTrials
VERUBULINSmall moleculeglioblastoma multiformeTubulin disrupting agent2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculelung cancerTubulin stabiliser3.0TerminatedClinicalTrials
ANG1005ProteinneoplasmTubulin inhibitor1.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeovarian mucinous adenocarcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
DOLASTATIN-10Small moleculelymphomaTubulin inhibitor2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculecolorectal cancerTubulin stabiliser1.0CompletedClinicalTrials
PLINABULINSmall moleculenon-small cell lung carcinomaTubulin inhibitor2.0Not yet recruitingClinicalTrials
MILATAXELSmall moleculemesotheliomaTubulin inhibitor2.0Unknown statusClinicalTrials
SOBLIDOTINSmall moleculeneoplasmTubulin inhibitor1.0WithdrawnClinicalTrials
PLINABULINSmall moleculeneutropeniaTubulin inhibitor3.0Active, not recruitingClinicalTrials
VINFLUNINESmall moleculeurinary bladder carcinomaTubulin inhibitor1.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculebreast cancerTubulin stabiliser1.0CompletedClinicalTrials
FOSBRETABULIN TROMETHAMINESmall moleculeovarian cancerTubulin disrupting agent2.0TerminatedClinicalTrials
ARX-788UnknowncancerTubulin inhibitor2.0WithdrawnClinicalTrials
FOSBRETABULINSmall moleculeneoplasmTubulin inhibitor2.0CompletedClinicalTrials
PLINABULINSmall moleculecancerTubulin inhibitor1.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeneoplasmTubulin stabiliser3.0-ATC
OMBRABULINSmall moleculeneoplasmTubulin inhibitor1.0CompletedClinicalTrials
ARX-788Unknownbreast neoplasmTubulin inhibitor2.0RecruitingClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodymalignant peripheral nerve sheath tumorTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculebreast cancerTubulin inhibitor2.0WithdrawnClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeprostate cancerTubulin stabiliser2.0TerminatedClinicalTrials
DOLASTATIN-10Small moleculemyelodysplastic syndromeTubulin inhibitor1.0CompletedClinicalTrials
OMBRABULINSmall moleculenon-small cell lung carcinomaTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculebladder transitional cell carcinomaTubulin inhibitor2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculebrain neoplasmTubulin stabiliser2.0CompletedClinicalTrials
SAGOPILONESmall moleculemelanomaTubulin stabiliser2.0CompletedClinicalTrials
FOSBRETABULIN TROMETHAMINESmall moleculeneuroendocrine neoplasmTubulin disrupting agent2.0CompletedClinicalTrials
DOLASTATIN-10Small moleculegallbladder cancerTubulin inhibitor2.0CompletedClinicalTrials
SAGOPILONESmall moleculesmall cell lung carcinomaTubulin stabiliser1.0CompletedClinicalTrials
DOLASTATIN-10Small moleculepancreatic carcinomaTubulin inhibitor2.0CompletedClinicalTrials
MILATAXELSmall moleculenon-small cell lung carcinomaTubulin inhibitor2.0CompletedClinicalTrials
LEXIBULINSmall moleculemultiple myelomaTubulin inhibitor2.0TerminatedClinicalTrials
VERUBULINSmall moleculebrain neoplasmTubulin disrupting agent1.0CompletedClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodysynovial sarcomaTubulin inhibitor2.0CompletedClinicalTrials
T-900607Small moleculeliver cancerTubulin disrupting agent2.0CompletedClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodyendometrial cancerTubulin inhibitor2.0RecruitingClinicalTrials
FOSBRETABULINSmall moleculeneoplasmTubulin inhibitor1.0CompletedClinicalTrials
VINFLUNINESmall moleculecancerTubulin inhibitor1.0WithdrawnClinicalTrials
ARX-788UnknownangiosarcomaTubulin inhibitor2.0RecruitingClinicalTrials
CROLIBULINSmall moleculecancerTubulin inhibitor1.0CompletedClinicalTrials
VINFLUNINESmall moleculeTransitional Cell CarcinomaTubulin inhibitor2.0Unknown statusClinicalTrials
ANG1005Proteinbrain neoplasmTubulin inhibitor2.0CompletedClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeOvarian Transitional Cell CarcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
VINFLUNINESmall moleculeneoplasmTubulin inhibitor1.0CompletedClinicalTrials
PLINABULINSmall moleculesmall cell lung carcinomaTubulin inhibitor1.0RecruitingClinicalTrials
SAGOPILONESmall moleculeCentral Nervous System NeoplasmTubulin stabiliser2.0CompletedClinicalTrials
DOLASTATIN-10Small moleculeleukemiaTubulin inhibitor1.0CompletedClinicalTrials
SAGOPILONESmall moleculebreast cancerTubulin stabiliser2.0CompletedClinicalTrials
ARX-788Unknownbreast cancerTubulin inhibitor2.0Active, not recruitingClinicalTrials
FOSBRETABULIN DISODIUMSmall moleculeneoplasmTubulin inhibitor1.0CompletedClinicalTrials
OMBRABULINSmall moleculesarcomaTubulin inhibitor3.0CompletedClinicalTrials
FOSBRETABULINSmall moleculehead and neck malignant neoplasiaTubulin inhibitor2.0CompletedClinicalTrials
VINFLUNINESmall moleculebreast cancerTubulin inhibitor2.0CompletedClinicalTrials
INDIBULINSmall moleculebreast cancerTubulin inhibitor1.0Unknown statusClinicalTrials
DOLASTATIN-10Small moleculeprostate cancerTubulin inhibitor2.0CompletedClinicalTrials
PLINABULINSmall moleculeneutropeniaTubulin inhibitor2.0CompletedClinicalTrials
LEXIBULINSmall moleculeglioblastoma multiformeTubulin inhibitor1.0TerminatedClinicalTrials
VINFLUNINESmall moleculegastric cancerTubulin inhibitor2.0TerminatedClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodybreast cancerTubulin inhibitor1.0WithdrawnClinicalTrials
PACLITAXEL POLIGLUMEXSmall moleculeendometrioid carcinomaTubulin stabiliser3.0Active, not recruitingClinicalTrials
INDIBULINSmall moleculeneoplasmTubulin inhibitor1.0Unknown statusClinicalTrials
INDIBULINSmall moleculeneoplasmTubulin inhibitor1.0CompletedClinicalTrials
SAGOPILONESmall moleculeovarian neoplasmTubulin stabiliser2.0CompletedClinicalTrials
PLINABULINSmall moleculeneutropeniaTubulin inhibitor3.0CompletedClinicalTrials
VINFLUNINESmall moleculeurinary bladder cancerTubulin inhibitor1.0WithdrawnClinicalTrials
MIRVETUXIMAB SORAVTANSINEAntibodybreast carcinomaTubulin inhibitor2.0CompletedClinicalTrials
PLINABULINSmall moleculenon-small cell lung carcinomaTubulin inhibitor1.0TerminatedClinicalTrials
LORVOTUZUMAB MERTANSINEAntibodyWilms tumorTubulin inhibitor2.0CompletedClinicalTrials