Drugs target to CDK9

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
DINACICLIBSmall moleculemultiple myelomaCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
SELICICLIBSmall moleculebreast cancerCyclin-dependent kinase 9 inhibitor1.0WithdrawnClinicalTrials
DINACICLIBSmall moleculeacute lymphoblastic leukemiaCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculeneoplasmCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
RONICICLIBSmall moleculesmall cell lung carcinomaCyclin-dependent kinase inhibitor2.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculeMantle cell lymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeendometrial cancerCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeprostate cancerCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculeacute myeloid leukemiaCyclin-dependent kinase 9 inhibitor1.0Active, not recruitingClinicalTrials
SELICICLIBSmall moleculenon-small cell lung carcinomaCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculenodal marginal zone B-cell lymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculeWaldenstrom macroglobulinemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculepancreatic adenocarcinomaCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeprolymphocytic leukemiaCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
BMS-387032Small moleculemultiple myelomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
RONICICLIBSmall moleculeneoplasmCyclin-dependent kinase inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeMALT lymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
PHA-793887Small moleculeneoplasmCyclin-dependent kinase inhibitor1.0TerminatedClinicalTrials
BMS-387032Small moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculesarcomaCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeesophageal cancerCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
DINACICLIBSmall moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor3.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeadult acute lymphoblastic leukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculemultiple myelomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculekidney cancerCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeliver cancerCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
DINACICLIBSmall moleculelentigo maligna melanomaCyclin-dependent kinase 9 inhibitor2.0Active, not recruitingClinicalTrials
ALVOCIDIBSmall moleculeSplenic Marginal Zone LymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
AT-7519Small moleculechronic lymphocytic leukemiaCyclin-dependent kinase inhibitor2.0CompletedClinicalTrials
DINACICLIBSmall moleculeneoplasmCyclin-dependent kinase 9 inhibitor1.0RecruitingClinicalTrials
ALVOCIDIBSmall moleculepancreatic adenocarcinomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeleukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
RONICICLIBSmall moleculesmall cell lung carcinomaCyclin-dependent kinase inhibitor1.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculemale breast carcinomaCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
ZOTIRACICLIBSmall moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculetherapy related acute myeloid leukemia and myelodysplastic syndromeCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculesmall intestine cancerCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculemultiple myelomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculeacral lentiginous melanomaCyclin-dependent kinase 9 inhibitor2.0Active, not recruitingClinicalTrials
ALVOCIDIBSmall moleculemyelodysplastic syndromeCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
DINACICLIBSmall moleculemucosal melanomaCyclin-dependent kinase 9 inhibitor2.0Active, not recruitingClinicalTrials
ALVOCIDIBSmall moleculeneoplasmCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculelymphoid neoplasmCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
SELICICLIBSmall moleculepituitary-dependent Cushing's diseaseCyclin-dependent kinase 9 inhibitor2.0Active, not recruitingClinicalTrials
RONICICLIBSmall moleculenon-small cell lung carcinomaCyclin-dependent kinase inhibitor1.0WithdrawnClinicalTrials
RGB-286638Small moleculelymphoid neoplasmCyclin-dependent kinase 9 inhibitor1.0WithdrawnClinicalTrials
ZOTIRACICLIBSmall moleculerectum cancerCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculefollicular lymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
SELICICLIBSmall moleculepituitary-dependent Cushing's diseaseCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculelymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculebreast cancerCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculemelanomaCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
BMS-387032Small moleculeneoplasmCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
AZD-5438Small moleculeneoplasmCyclin-dependent kinase inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculeacute myeloid leukemiaCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
SELICICLIBSmall moleculeneoplasmCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
RONICICLIBSmall moleculeneoplasmCyclin-dependent kinase inhibitor2.0WithdrawnClinicalTrials
BMS-387032Small moleculeMantle cell lymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculebreast cancerCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculecutaneous melanomaCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
AT-7519Small moleculeneoplasmCyclin-dependent kinase inhibitor1.0Active, not recruitingClinicalTrials
ZOTIRACICLIBSmall moleculehepatocellular carcinomaCyclin-dependent kinase 9 inhibitor1.0WithdrawnClinicalTrials
ALVOCIDIBSmall moleculeacute myeloid leukemiaCyclin-dependent kinase 9 inhibitor1.0WithdrawnClinicalTrials
AT-7519Small moleculemultiple myelomaCyclin-dependent kinase inhibitor1.0CompletedClinicalTrials
SELICICLIBSmall moleculecystic fibrosisCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
ZOTIRACICLIBSmall moleculeglioblastoma multiformeCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ZOTIRACICLIBSmall moleculegliosarcomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeprolymphocytic leukemiaCyclin-dependent kinase 9 inhibitor1.0TerminatedClinicalTrials
ALVOCIDIBSmall moleculechronic lymphocytic leukemiaCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
ALVOCIDIBSmall moleculemultiple myelomaCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
ALVOCIDIBSmall moleculediffuse large B-cell lymphomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeacute myeloid leukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculeprolymphocytic leukemiaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeprostate cancerCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials
AT-7519Small moleculelymphomaCyclin-dependent kinase inhibitor1.0CompletedClinicalTrials
DINACICLIBSmall moleculepancreatic adenocarcinomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculecutaneous melanomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
ALVOCIDIBSmall moleculeacute myeloid leukemiaCyclin-dependent kinase 9 inhibitor2.0TerminatedClinicalTrials
DINACICLIBSmall moleculemale breast carcinomaCyclin-dependent kinase 9 inhibitor1.0CompletedClinicalTrials
AT-7519Small moleculeMantle cell lymphomaCyclin-dependent kinase inhibitor2.0CompletedClinicalTrials
ALVOCIDIBSmall moleculelymphomaCyclin-dependent kinase 9 inhibitor2.0CompletedClinicalTrials