Drugs target to THRA

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0RecruitingClinicalTrials
LIOTHYRONINE SODIUMSmall moleculethyroid neoplasmThyroid hormone receptor agonist2.0CompletedClinicalTrials
LIOTHYRONINE SODIUMSmall moleculecongenital heart diseaseThyroid hormone receptor agonist3.0Unknown statusClinicalTrials
LIOTHYRONINE SODIUMSmall moleculemyxedemaThyroid hormone receptor agonist4.0-DailyMed
DEXTROTHYROXINESmall moleculemyocardial infarctionThyroid hormone receptor agonist3.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist2.0Active, not recruitingClinicalTrials
LIOTHYRONINESmall moleculedepressive disorderThyroid hormone receptor agonist4.0TerminatedClinicalTrials
LEVOTHYROXINESmall moleculethyroid cancerThyroid hormone receptor agonist4.0TerminatedClinicalTrials
LIOTHYRONINESmall moleculeseptic shockThyroid hormone receptor agonist2.0RecruitingClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculehypothyroidismThyroid hormone receptor agonist4.0Unknown statusClinicalTrials
LEVOTHYROXINESmall moleculebipolar disorderThyroid hormone receptor agonist2.0CompletedClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculethyroid carcinomaThyroid hormone receptor agonist4.0-DailyMed
LIOTHYRONINESmall moleculemyxedemaThyroid hormone receptor agonist4.0-DailyMed
LEVOTHYROXINESmall moleculethyroid carcinomaThyroid hormone receptor agonist4.0-DailyMed
LEVOTHYROXINE SODIUMSmall moleculehypothyroidismThyroid hormone receptor agonist2.0CompletedClinicalTrials
LIOTHYRONINE SODIUMSmall moleculeprostate cancerThyroid hormone receptor agonist1.0TerminatedClinicalTrials
LIOTHYRONINESmall moleculechronic progressive multiple sclerosisThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculehead and neck malignant neoplasiaThyroid hormone receptor agonist1.0RecruitingClinicalTrials
LEVOTHYROXINESmall moleculeGraves diseaseThyroid hormone receptor agonist2.0CompletedClinicalTrials
DEXTROTHYROXINE SODIUMSmall moleculeMyocardial IschemiaThyroid hormone receptor agonist3.0CompletedClinicalTrials
DEXTROTHYROXINESmall moleculeDown syndromeThyroid hormone receptor agonist3.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculegoiterThyroid hormone receptor agonist4.0WithdrawnClinicalTrials
LEVOTHYROXINESmall moleculecongenital hypothyroidismThyroid hormone receptor agonist3.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0-DailyMed
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0WithdrawnClinicalTrials
LIOTHYRONINESmall moleculedifferentiated thyroid carcinomaThyroid hormone receptor agonist4.0-DailyMed
LEVOTHYROXINESmall moleculethyroid cancerThyroid hormone receptor agonist4.0-DailyMed
LIOTHYRONINESmall moleculebreast cancerThyroid hormone receptor agonist2.0TerminatedClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist2.0CompletedClinicalTrials
LIOTHYRONINESmall moleculedepressive disorderThyroid hormone receptor agonist3.0CompletedClinicalTrials
LIOTHYRONINESmall moleculeatrial fibrillationThyroid hormone receptor agonist1.0CompletedClinicalTrials
LIOTHYRONINESmall moleculeAbnormality of cardiovascular system morphologyThyroid hormone receptor agonist1.0CompletedClinicalTrials
LIOTHYRONINESmall moleculeunipolar depressionThyroid hormone receptor agonist3.0CompletedClinicalTrials
LIOTHYRONINESmall moleculehypothyroidismThyroid hormone receptor agonist2.0CompletedClinicalTrials
LIOTHYRONINESmall moleculehead and neck malignant neoplasiaThyroid hormone receptor agonist1.0CompletedClinicalTrials
LIOTHYRONINE SODIUMSmall moleculehead and neck malignant neoplasiaThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculehypothyroidismThyroid hormone receptor agonist4.0CompletedClinicalTrials
LIOTHYRONINE SODIUMSmall moleculedifferentiated thyroid carcinomaThyroid hormone receptor agonist4.0-DailyMed
LIOTHYRONINESmall moleculebipolar disorderThyroid hormone receptor agonist3.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0TerminatedClinicalTrials
LEVOTHYROXINESmall moleculepainThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculepregnancyThyroid hormone receptor agonist0.5Unknown statusClinicalTrials
LIOTHYRONINESmall moleculeprostate cancerThyroid hormone receptor agonist1.0TerminatedClinicalTrials
LIOTHYRONINESmall moleculedepressive disorderThyroid hormone receptor agonist4.0CompletedClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculedifferentiated thyroid carcinomaThyroid hormone receptor agonist4.0-DailyMed
LIOTHYRONINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0-DailyMed
LEVOTHYROXINE SODIUMSmall moleculehypothyroidismThyroid hormone receptor agonist4.0RecruitingClinicalTrials
LEVOTHYROXINESmall moleculecongenital hypothyroidismThyroid hormone receptor agonist4.0RecruitingClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculebipolar disorderThyroid hormone receptor agonist2.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculediabetes mellitusThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculedifferentiated thyroid carcinomaThyroid hormone receptor agonist4.0-DailyMed
LIOTHYRONINESmall moleculegliosarcomaThyroid hormone receptor agonist0.5WithdrawnClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculepainThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculeDisorder of lipid metabolismThyroid hormone receptor agonist3.0Unknown statusClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculethyroid cancerThyroid hormone receptor agonist4.0-DailyMed
LEVOTHYROXINESmall moleculesystemic lupus erythematosusThyroid hormone receptor agonist4.0WithdrawnClinicalTrials
DEXTROTHYROXINE SODIUMSmall moleculemyocardial infarctionThyroid hormone receptor agonist3.0CompletedClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculehypothyroidismThyroid hormone receptor agonist4.0-DailyMed
LIOTHYRONINE SODIUMSmall moleculeAbnormality of cardiovascular system morphologyThyroid hormone receptor agonist3.0CompletedClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculenodular goiterThyroid hormone receptor agonist4.0CompletedClinicalTrials
LIOTHYRONINE SODIUMSmall moleculemultiple sclerosisThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist0.5CompletedClinicalTrials
LIOTHYRONINESmall moleculemultiple sclerosisThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculecongenital hypothyroidismThyroid hormone receptor agonist4.0CompletedClinicalTrials
DEXTROTHYROXINESmall moleculecardiovascular diseaseThyroid hormone receptor agonist4.0-ATC
LIOTHYRONINESmall moleculeAbnormality of cardiovascular system morphologyThyroid hormone receptor agonist3.0CompletedClinicalTrials
LIOTHYRONINESmall moleculethyroid neoplasmThyroid hormone receptor agonist2.0CompletedClinicalTrials
LIOTHYRONINE SODIUMSmall moleculehypothyroidismThyroid hormone receptor agonist4.0-DailyMed
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0Unknown statusClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculecongenital hypothyroidismThyroid hormone receptor agonist4.0-DailyMed
LIOTHYRONINESmall moleculeeuthyroid sick syndromeThyroid hormone receptor agonist2.0RecruitingClinicalTrials
LIOTHYRONINESmall moleculecongenital heart diseaseThyroid hormone receptor agonist3.0Unknown statusClinicalTrials
LEVOTHYROXINESmall moleculenodular goiterThyroid hormone receptor agonist4.0CompletedClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculecongenital hypothyroidismThyroid hormone receptor agonist4.0RecruitingClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist3.0RecruitingClinicalTrials
LIOTHYRONINESmall moleculeheart failureThyroid hormone receptor agonist1.0RecruitingClinicalTrials
LEVOTHYROXINE SODIUMSmall moleculehead and neck malignant neoplasiaThyroid hormone receptor agonist1.0RecruitingClinicalTrials
LEVOTHYROXINESmall moleculeeuthyroid sick syndromeThyroid hormone receptor agonist4.0CompletedClinicalTrials
LIOTHYRONINESmall moleculerelapsing-remitting multiple sclerosisThyroid hormone receptor agonist1.0CompletedClinicalTrials
LEVOTHYROXINESmall moleculehypothyroidismThyroid hormone receptor agonist4.0Active, not recruitingClinicalTrials
LEVOTHYROXINESmall moleculecongenital hypothyroidismThyroid hormone receptor agonist4.0-DailyMed
DEXTROTHYROXINESmall moleculeMyocardial IschemiaThyroid hormone receptor agonist3.0CompletedClinicalTrials