Drugs target to MAPK14

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
LOSMAPIMODSmall moleculeFacioscapulohumeral dystrophyMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
ARRY-797Small moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
ARRY-797Small moleculeankylosing spondylitisMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
DORAMAPIMODSmall moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
PH-797804Small moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
TALMAPIMODSmall moleculemultiple myelomaMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
FX-005Small moleculeosteoarthritis, kneeMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
TAK-715Small moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
RALIMETINIBSmall moleculeovarian cancerMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
RALIMETINIBSmall moleculeprimary peritoneal carcinomaMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeCOVID-19MAP kinase p38 alpha inhibitor3.0TerminatedClinicalTrials
ARRY-797Small moleculeosteoarthritis, kneeMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
PEXMETINIBSmall moleculemyelodysplastic syndromeMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
PF-03715455Small moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
LOSMAPIMODSmall moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
NEFLAMAPIMODSmall moleculeDementiaMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
RALIMETINIBSmall moleculecancerMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
NEFLAMAPIMODSmall moleculeHuntington diseaseMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
NEFLAMAPIMODSmall moleculeAlzheimer diseaseMAP kinase p38 alpha inhibitor2.0RecruitingClinicalTrials
PH-797804Small moleculepostherpetic neuralgiaMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeatherosclerosisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
ARRY-797Small moleculedilated cardiomyopathyMAP kinase p38 alpha inhibitor3.0Active, not recruitingClinicalTrials
PH-797804Small moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeatherosclerosisMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
DORAMAPIMODSmall moleculepsoriasisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeacute coronary syndromeMAP kinase p38 alpha inhibitor3.0CompletedClinicalTrials
SEMAPIMODSmall moleculeCrohn's diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
PH-797804Small moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculefocal segmental glomerulosclerosisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
NEFLAMAPIMODSmall moleculeAlzheimer diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
RALIMETINIBSmall moleculeglioblastoma multiformeMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculecardiovascular diseaseMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
PF-03715455Small moleculeasthmaMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
DILMAPIMODSmall moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculemajor depressive disorderMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeFacioscapulohumeral dystrophyMAP kinase p38 alpha inhibitor2.0Active, not recruitingClinicalTrials
BMS-582949Small moleculepsoriasisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
PG-760564Small moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
TALMAPIMODSmall moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
GSK-610677Small moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculemajor depressive disorderMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
DILMAPIMODSmall moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
SEMAPIMODSmall moleculeCrohn's diseaseMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
DILMAPIMODSmall moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
RALIMETINIBSmall moleculefallopian tube cancerMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeacute coronary syndromeMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
ARRY-797Small moleculetoothacheMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
DILMAPIMODSmall moleculeacute lung injuryMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
AZD-7624Small moleculeinflammationMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
PH-797804Small moleculeosteoarthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
ACUMAPIMODSmall moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeFacioscapulohumeral dystrophyMAP kinase p38 alpha inhibitor3.0RecruitingClinicalTrials
ARRY-797Small moleculedilated cardiomyopathyMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
PH-797804Small moleculepainMAP kinase p38 alpha inhibitor1.0WithdrawnClinicalTrials
DILMAPIMODSmall moleculeneuropathic painMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
AZD-7624Small moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
DILMAPIMODSmall moleculecoronary artery diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
AZD-7624Small moleculeasthmaMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
TALMAPIMODSmall moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LY-3007113Small moleculemetastatic malignant neoplasmMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeneuropathic painMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
AZD-7624Small moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
VX-702Small moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
KC-706Small moleculepemphigus vulgarisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
PF-03715455Small moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials
RALIMETINIBSmall moleculebreast cancerMAP kinase p38 alpha inhibitor2.0TerminatedClinicalTrials
DILMAPIMODSmall moleculechronic obstructive pulmonary diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
BMS-582949Small moleculerheumatoid arthritisMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
NEFLAMAPIMODSmall moleculeCognitive impairmentMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
BMS-582949Small moleculevascular diseaseMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeDisorder of lipid metabolismMAP kinase p38 alpha inhibitor2.0CompletedClinicalTrials
LOSMAPIMODSmall moleculeacute coronary syndromeMAP kinase p38 alpha inhibitor1.0CompletedClinicalTrials