Drugs target to EZH2

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
TAZEMETOSTAT HYDROBROMIDESmall moleculefollicular lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor4.0-DailyMed
TAZEMETOSTATSmall moleculeurothelial carcinomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculemultiple myelomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculefollicular lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor3.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculeurinary bladder cancerHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculenasal cavity and paranasal sinus carcinomaHistone-lysine N-methyltransferase EZH2 inhibitor2.0Not yet recruitingClinicalTrials
TAZEMETOSTATSmall moleculeprostate cancerHistone-lysine N-methyltransferase EZH2 inhibitor0.5Not yet recruitingClinicalTrials
TAZEMETOSTATSmall moleculemesotheliomaHistone-lysine N-methyltransferase EZH2 inhibitor2.0CompletedClinicalTrials
TAZEMETOSTAT HYDROBROMIDESmall moleculesarcomaHistone-lysine N-methyltransferase EZH2 inhibitor4.0-FDA
TAZEMETOSTATSmall moleculehead and neck squamous cell carcinomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculesmall cell lung carcinomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculefollicular lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor2.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculefollicular lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculenon-Hodgkins lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculesarcomaHistone-lysine N-methyltransferase EZH2 inhibitor4.0-FDA
TAZEMETOSTATSmall moleculediffuse large B-cell lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculenon-small cell lung carcinomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0Not yet recruitingClinicalTrials
TAZEMETOSTATSmall moleculefollicular lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0Not yet recruitingClinicalTrials
TAZEMETOSTATSmall moleculeacute myeloid leukemiaHistone-lysine N-methyltransferase EZH2 inhibitor1.0Not yet recruitingClinicalTrials
TAZEMETOSTATSmall moleculeneoplasm of mature B-cellsHistone-lysine N-methyltransferase EZH2 inhibitor1.0CompletedClinicalTrials
TAZEMETOSTATSmall moleculefollicular lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor4.0-DailyMed
TAZEMETOSTATSmall moleculediffuse large B-cell lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0Not yet recruitingClinicalTrials
TAZEMETOSTATSmall moleculelymphomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0CompletedClinicalTrials
TAZEMETOSTATSmall moleculemetastatic prostate cancerHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculeepithelioid sarcomaHistone-lysine N-methyltransferase EZH2 inhibitor3.0RecruitingClinicalTrials
GSK2816126Small moleculecancerHistone-lysine N-methyltransferase EZH2 inhibitor1.0TerminatedClinicalTrials
TAZEMETOSTATSmall moleculefollicular lymphomaHistone-lysine N-methyltransferase EZH2 inhibitor2.0TerminatedClinicalTrials
TAZEMETOSTATSmall moleculeneoplasmHistone-lysine N-methyltransferase EZH2 inhibitor2.0RecruitingClinicalTrials
TAZEMETOSTAT HYDROBROMIDESmall moleculeprostate cancerHistone-lysine N-methyltransferase EZH2 inhibitor0.5Not yet recruitingClinicalTrials
TAZEMETOSTAT HYDROBROMIDESmall moleculesmall cell lung carcinomaHistone-lysine N-methyltransferase EZH2 inhibitor1.0RecruitingClinicalTrials
TAZEMETOSTATSmall moleculeneoplasmHistone-lysine N-methyltransferase EZH2 inhibitor4.0-ATC
TAZEMETOSTATSmall moleculeneoplasm of mature B-cellsHistone-lysine N-methyltransferase EZH2 inhibitor2.0CompletedClinicalTrials