Drugs target to HSP90AA1

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
TANESPIMYCINSmall moleculeanaplastic large cell lymphomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
BIIB021Small moleculebreast cancerHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculelung cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
SNX 5422Small moleculelymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculelung cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculemedullary thyroid gland carcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
GANETESPIBSmall moleculesmall cell lung carcinomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculenodal marginal zone B-cell lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeBurkitts lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculebreast cancerHeat shock protein HSP90 inhibitor1.0WithdrawnClinicalTrials
RETASPIMYCINSmall moleculeprostate adenocarcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculecancerHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
ALVESPIMYCINSmall moleculebreast cancerHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
GANETESPIBSmall moleculerectum cancerHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculecentral nervous system non-hodgkin lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculemelanomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
GANETESPIBSmall moleculefallopian tube cancerHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculebreast cancerHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
GANETESPIBSmall moleculeangiosarcomaHeat shock protein HSP90 inhibitor2.0RecruitingClinicalTrials
BIIB021Small moleculechronic lymphocytic leukemiaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculegastrointestinal stromal tumorHeat shock protein HSP90 inhibitor3.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculemultiple myelomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
GANETESPIBSmall moleculemelanomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeMantle cell lymphomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeMantle cell lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculefollicular lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
SNX 5422Small moleculecancerHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeovarian sarcomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
BIIB021Small moleculeneoplasmHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeosteosarcomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculechronic myeloproliferative disorderHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeHodgkins lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculekidney cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCINSmall moleculelung cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeLymphoma, AIDS-RelatedHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculelymphoblastic lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculegastric cancerHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
LUMINESPIBSmall moleculegastrointestinal stromal tumorHeat shock protein HSP90 inhibitor2.0Unknown statusClinicalTrials
GANETESPIBSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeangioimmunoblastic T-cell lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeprolymphocytic leukemiaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculefollicular lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
LUMINESPIBSmall moleculegastric cancerHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
BIIB021Small moleculebreast cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
SNX 5422Small moleculeleukemiaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculemalignant colon neoplasmHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ONALESPIBSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculelymphoblastic lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculemycosis fungoidesHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeadult T-cell leukemia/lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculehead and neck malignant neoplasiaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculehepatocellular carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ONALESPIBSmall moleculebreast carcinomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
LUMINESPIBSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculebreast cancerHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculebreast carcinomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeBurkitts lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
CD24FCUnknownmetastatic melanomaHeat shock protein HSP90 inhibitor1.0WithdrawnClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculeprostate adenocarcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculepapillary thyroid carcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeanaplastic large cell lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
GANETESPIBSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
CD24FCUnknownCOVID-19Heat shock protein HSP90 inhibitor3.0CompletedClinicalTrials
SNX 5422Small moleculehematopoietic and lymphoid cell neoplasmHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ALVESPIMYCINSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0Unknown statusClinicalTrials
LUMINESPIBSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeWaldenstrom macroglobulinemiaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
GANETESPIBSmall moleculeovarian cancerHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculelymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculemultiple myelomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculemultiple myelomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCINSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculechronic lymphocytic leukemiaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCINSmall moleculelung cancerHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculelung cancerHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculemycosis fungoidesHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculebreast cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ALVESPIMYCINSmall moleculebreast cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculenodal marginal zone B-cell lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
SNX 5422Small moleculecancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculemelanomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculediffuse large B-cell lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculelymphomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
LUMINESPIBSmall moleculerectum cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeHodgkins lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeangioimmunoblastic T-cell lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculemalignant peripheral nerve sheath tumorHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculegastroesophageal junction adenocarcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculeprimary peritoneal carcinomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
GANETESPIBSmall moleculemalignant colon neoplasmHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculecutaneous melanomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
CD24FCUnknownneoplasmHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeEwing sarcoma/peripheral primitive neuroectodermal tumorHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculepancreatic adenocarcinomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
RETASPIMYCINSmall moleculemetastatic melanomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculecutaneous melanomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculelung adenocarcinomaHeat shock protein HSP90 inhibitor3.0TerminatedClinicalTrials
GANETESPIBSmall moleculegastrointestinal stromal tumorHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculecolorectal carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculesmall intestine lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeHodgkins lymphomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
GANETESPIBSmall moleculesmall cell lung carcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculelymphomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeLymphoma, AIDS-RelatedHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculemultiple myelomaHeat shock protein HSP90 inhibitor3.0CompletedClinicalTrials
GANETESPIBSmall moleculemale breast carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculemultiple myelomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculebreast cancerHeat shock protein HSP90 inhibitor1.0WithdrawnClinicalTrials
TANESPIMYCINSmall moleculegastric cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeleukemiaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
LUMINESPIBSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculemetastatic melanomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeanaplastic large cell lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCINSmall moleculededifferentiated liposarcomaHeat shock protein HSP90 inhibitor2.0WithdrawnClinicalTrials
TANESPIMYCINSmall moleculediffuse large B-cell lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
GANETESPIBSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0Unknown statusClinicalTrials
GANETESPIBSmall moleculeesophageal carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ONALESPIBSmall moleculebreast cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ONALESPIBSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0Active, not recruitingClinicalTrials
LUMINESPIBSmall moleculemyeloproliferative disorderHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
RETASPIMYCINSmall moleculebreast cancerHeat shock protein HSP90 inhibitor1.0WithdrawnClinicalTrials
TANESPIMYCINSmall moleculechronic lymphocytic leukemiaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeMALT lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ONALESPIBSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor1.0Active, not recruitingClinicalTrials
TANESPIMYCINSmall moleculepancreatic adenocarcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeSplenic Marginal Zone LymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculekidney cancerHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeSezary's diseaseHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculebreast cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculeprostate adenocarcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
GANETESPIBSmall moleculetriple-negative breast cancerHeat shock protein HSP90 inhibitor2.0RecruitingClinicalTrials
TANESPIMYCINSmall moleculecancerHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
GANETESPIBSmall moleculeacute myeloid leukemiaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeprostate adenocarcinomaHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
ALVESPIMYCINSmall moleculeprolymphocytic leukemiaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
RETASPIMYCINSmall moleculemultiple myelomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculededifferentiated liposarcomaHeat shock protein HSP90 inhibitor2.0WithdrawnClinicalTrials
TANESPIMYCINSmall moleculeurinary bladder cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculemyelodysplastic syndromeHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ALVESPIMYCINSmall moleculechronic lymphocytic leukemiaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
GANETESPIBSmall moleculegastric cancerHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeSezary's diseaseHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
BIIB021Small moleculelymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculemalignant pleural mesotheliomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculechondrosarcomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
SNX 5422Small moleculecancerHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
LUMINESPIBSmall moleculelung adenocarcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ONALESPIBSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeMALT lymphomaHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
GANETESPIBSmall moleculeneoplasmHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
GANETESPIBSmall moleculelung cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCINSmall moleculegastrointestinal stromal tumorHeat shock protein HSP90 inhibitor3.0TerminatedClinicalTrials
LUMINESPIBSmall moleculecolorectal adenocarcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeovarian cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeprostate cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCIN HYDROCHLORIDESmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculerectum cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCINSmall moleculecancerHeat shock protein HSP90 inhibitor1.0TerminatedClinicalTrials
LUMINESPIBSmall moleculegastrointestinal stromal tumorHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeadult T-cell leukemia/lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeleukemiaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
GANETESPIBSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
RETASPIMYCINSmall moleculebreast carcinomaHeat shock protein HSP90 inhibitor2.0TerminatedClinicalTrials
TANESPIMYCINSmall moleculeMantle cell lymphomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
LUMINESPIBSmall moleculesquamous cell lung carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
ONALESPIBSmall moleculeprostate cancerHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
TANESPIMYCINSmall moleculeuterine sarcomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
RETASPIMYCINSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials
BIIB021Small moleculegastrointestinal stromal tumorHeat shock protein HSP90 inhibitor2.0CompletedClinicalTrials
LUMINESPIBSmall moleculenon-small cell lung carcinomaHeat shock protein HSP90 inhibitor1.0CompletedClinicalTrials