Drugs target to POLR1A

Drug name Drug type Disease/phenotype Mechanism of action(MoA) Phase Status Source
TAS-106Small moleculecancerDNA-directed RNA polymerase I subunit RPA1 inhibitor1.0CompletedClinicalTrials
TAS-106Small moleculehead and neck malignant neoplasiaDNA-directed RNA polymerase I subunit RPA1 inhibitor2.0TerminatedClinicalTrials